Table 1. Pharmacokinetic Parameters following Intramuscular Administration of Trelstar Depot to Healthy Male Volunteers

DESCRIPTION TRELSTAR  DEPOT contains a pamoate salt of triptorelin, and triptorelin is a synthetic decapeptide agonist analog of luteinizing hormone releasing hormone (LHRH or GnRH) with greater potency than the naturally occurring LHRH. The chemical name of triptorelin pamoate is 5-oxo-L-prolyl-L-histidyl-L-tryptophyl-L-serylL-tyrosyl-D-tryptophyl-L-leucyl-L-arginyl-L-prolylglycine amide (pamoate salt); the empirical formula is C64H82N18O13 · C23H16O6 and the molecular weight is 1699.9. The structural formula is shown below.